SCHEMBL7313890

SCHEMBL7313890

CCCC[C@H](NC(=O)CCCCNC(=O)COc1ccc(C)cc1)C(=O)C[S@@+]([O-])Cc1ccco1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
TSHR P16473 2/20 0.42
MAPK1 P28482 2/20 0.42
PKM P14618 1/20 0.42
ALDH1A1 P00352 9/20 0.42
POLB P06746 2/20 0.42
MAPT P10636 3/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RECQL P46063 2/20 0.38
TRPM8 Q7Z2W7 1/20 0.38
LMNA P02545 1/20 0.38
HDAC1 Q13547 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
USP2 O75604 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7302470 0.84 ALDH1A1 (0.49) HPGDCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7307300 0.84 TSHR (0.45) HPGDCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7313905 0.83 PKM (0.41) HPGDCYP1A2CYP2C9CYP2C19TSHR
SCHEMBL7311204 0.80 ALDH1A1 (0.49) HPGDCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7313884 0.78 CASP3 (0.44) HPGDPKMALDH1A1POLBMAPT
SCHEMBL7313900 0.78 CASP3 (0.44) HPGDPKMALDH1A1POLBMAPT
SCHEMBL7301633 0.75 ALDH1A1 (0.51) HPGDCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7303788 0.73 ALDH1A1 (0.52) HPGDCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7312907 0.72 HPGD (0.48) HPGDCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7315648 0.72 ALDH1A1 (0.51) HPGDCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed