SCHEMBL7313900

SCHEMBL7313900

CCCCC(NC(=O)C(CC(C)C)NC(=O)COc1ccccc1)C(=O)C[S+]([O-])Cc1ccco1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 8/20 0.44
CASP1 P29466 7/20 0.42
CASP7 P55210 7/20 0.42
CASP6 P55212 6/20 0.42
CASP8 Q14790 6/20 0.42
CTSD P07339 1/20 0.40
REN P00797 1/20 0.39
PKM P14618 1/20 0.38
ALDH1A1 P00352 3/20 0.38
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
MMP9 P14780 1/20 0.38
USP2 O75604 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PSMB5 P28074 1/20 0.37
CAPNS1 P04632 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313884 1.00 CASP3 (0.44) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7313905 0.84 PKM (0.41) PKMALDH1A1USP2POLBMAPT
SCHEMBL7302479 0.84 ALDH1A1 (0.48) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7302463 0.84 ALDH1A1 (0.48) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7307309 0.83 CASP3 (0.45) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7307297 0.83 CASP3 (0.45) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7311213 0.79 ALDH1A1 (0.49) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7311200 0.79 ALDH1A1 (0.49) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7313890 0.78 HPGD (0.44) PKMALDH1A1USP2POLBMAPT
SCHEMBL7313893 0.78 MAPT (0.36) PKMALDH1A1USP2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed