SCHEMBL7315407

SCHEMBL7315407

COC(=O)CCc1c(O)nc(C)c2c(OC)c(OC)c(OC)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
DPP4 P27487 2/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
ATM Q13315 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
BACE1 P56817 1/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36
TUBB8 Q3ZCM7 1/20 0.36
TUBA3E Q6PEY2 1/20 0.36
TUBA1A Q71U36 1/20 0.36
TUBA1C Q9BQE3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7305966 0.84 PDE3B (0.57) PDE3BPDE3AGAABACE1TSHR
SCHEMBL7307946 0.76 PDE3B (0.54) PDE3BPDE3ABACE1TSHRKDM4E
SCHEMBL7319852 0.75 HPGD (0.37) MAPTALDH1A1KMT2AKDM4EMEN1
Perchlorate SCHEMBL7312607 0.73 PDE3B (0.43) PDE3BPDE3ADPP4NPC1GAA
SCHEMBL7311043 0.73 PDE3B (0.50) PDE3BPDE3ADPP4NPC1BACE1
SCHEMBL7315403 0.72 SLC10A2 (0.37) DPP4GAATUBB4ATUBBTUBA3C
SCHEMBL7313861 0.72 PDE3B (0.44) PDE3BPDE3ADPP4GAAMAPT
SCHEMBL7317446 0.72 TP53 (0.44) PDE3BPDE3AMAPTALDH1A1KDM4E
SCHEMBL7309250 0.70 PDE3B (0.44) PDE3BPDE3ADPP4GAATSHR
SCHEMBL7319613 0.70 ALDH1A1 (0.41) PDE3BPDE3ANPC1ATMRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4822800-A Isoquinolinol compounds having cardiotonic and phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-04-18 US disclosed