SCHEMBL7315508

SCHEMBL7315508

CC(S)Cc1ncnc(O)c1Cc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.42
ALDH1A1 P00352 5/20 0.39
CYP1A2 P05177 5/20 0.39
CYP3A4 P08684 5/20 0.39
HSD17B10 Q99714 5/20 0.39
CLK4 Q9HAZ1 3/20 0.39
MAPK1 P28482 2/20 0.39
MME P08473 1/20 0.37
FFAR1 O14842 1/20 0.37
AKR1B1 P15121 1/20 0.37
HPGD P15428 2/20 0.36
BRS3 P32247 2/20 0.36
PTPN1 P18031 1/20 0.36
CYP2C9 P11712 2/20 0.36
TSHR P16473 2/20 0.36
CYP2C19 P33261 2/20 0.36
GSK3A P49840 2/20 0.36
GSK3B P49841 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9308863 0.84 PPARG (0.46) ESR2ALDH1A1CYP1A2CYP3A4HSD17B10
SCHEMBL9846002 0.82 ACHE (0.43) ESR2ALDH1A1CYP1A2CYP3A4HSD17B10
SCHEMBL9309571 0.73 ESR2 (0.45) ESR2MMEFFAR1AKR1B1GSK3A
SCHEMBL8312740 0.72 PPARG (0.48) ESR2PPARG
SCHEMBL9310919 0.72 PPARG (0.47) ESR2ALDH1A1CYP1A2CYP3A4HSD17B10
SCHEMBL2843118 0.72 BRS3 (0.38) ESR2MMEFFAR1AKR1B1BRS3
SCHEMBL9846033 0.71 PPARG (0.43) ESR2PPARG
SCHEMBL9311025 0.71 PPARG (0.49) ESR2FFAR1AKR1B1PPARG
SCHEMBL9307715 0.71 PPARG (0.49) ESR2PPARG
SCHEMBL9309735 0.70 PPARG (0.48) ESR2FFAR1AKR1B1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5231094-A Cardiovascular disorders SOCIETE ANONYME: LABORATOIRES UPSA (FR) 1993-07-27 US disclosed