SCHEMBL9846002

SCHEMBL9846002

CCCCc1ncnc(O)c1Cc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.43
ESR2 Q92731 1/20 0.43
PPARG P37231 2/20 0.42
AGTR1 P30556 2/20 0.41
APLNR P35414 1/20 0.40
FFAR1 O14842 1/20 0.40
AKR1B1 P15121 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
AGTR2 P50052 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9308863 0.93 PPARG (0.46) ACHEESR2PPARGFFAR1AKR1B1
SCHEMBL9308844 0.85 PPARG (0.45) ACHEESR2PPARGAGTR1APLNR
SCHEMBL9846039 0.85 PPARG (0.45) ACHEESR2PPARGAGTR1APLNR
SCHEMBL9846092 0.84 PPARG (0.45) ACHEESR2PPARGAGTR1APLNR
SCHEMBL9846024 0.84 PPARG (0.47) ACHEESR2PPARGAGTR1APLNR
SCHEMBL9846033 0.83 PPARG (0.43) ACHEESR2PPARGAGTR1APLNR
SCHEMBL7315508 0.82 ESR2 (0.42) ESR2PPARGFFAR1AKR1B1ALDH1A1
SCHEMBL9310919 0.81 PPARG (0.47) ACHEESR2PPARGAGTR1FFAR1
SCHEMBL8979828 0.80 ACHE (0.46) ACHEPPARGAGTR1
SCHEMBL9308992 0.79 CYP1A2 (0.45) ACHEESR2PPARGFFAR1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0424317-A2 Pyrimidines CIBA-GEIGY AG (CH) 1991-04-24 EP disclosed