SCHEMBL7315524

SCHEMBL7315524

O=S(=O)(c1cccc2cnccc12)N1CCCC(O)C1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.62
PRKD3 O94806 3/20 0.62
PRKCG P05129 3/20 0.62
PRKCB P05771 3/20 0.62
PRKCA P17252 3/20 0.62
PRKCH P24723 3/20 0.62
PRKCI P41743 3/20 0.62
PRKCE Q02156 3/20 0.62
PRKCQ Q04759 3/20 0.62
PRKCZ Q05513 3/20 0.62
PRKCD Q05655 3/20 0.62
PRKD1 Q15139 3/20 0.62
CYP2D6 P10635 2/20 0.62
NFKB1 P19838 1/20 0.62
ROCK2 O75116 11/20 0.61
ROCK1 Q13464 10/20 0.61
CCR2 P41597 2/20 0.61
ADORA3 P0DMS8 2/20 0.61
PRKACA P17612 2/20 0.61
PRKACG P22612 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7326564 0.93 ROCK2 (0.65) CYP3A4PRKD3PRKCGPRKCBPRKCA
SCHEMBL4728844 0.86 ROCK2 (0.62) CYP3A4PRKD3PRKCGPRKCBPRKCA
SCHEMBL7318375 0.85 ROCK2 (0.71) CYP3A4PRKD3PRKCGPRKCBPRKCA
SCHEMBL4727734 0.85 CYP3A4 (0.62) CYP3A4PRKD3PRKCGPRKCBPRKCA
SCHEMBL4705021 0.85 MEN1 (0.65) MEN1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL9194379 0.85 ROCK2 (0.62) CYP3A4PRKD3PRKCGPRKCBPRKCA
SCHEMBL10988523 0.84 ROCK2 (0.79) CYP3A4PRKD3PRKCGPRKCBPRKCA
SCHEMBL4726515 0.83 ROCK2 (0.68) CYP3A4PRKD3PRKCGPRKCBPRKCA
SCHEMBL4727367 0.83 CYP3A4 (0.62) CYP3A4PRKD3PRKCGPRKCBPRKCA
SCHEMBL10985139 0.82 ROCK2 (0.77) CYP3A4PRKD3PRKCGPRKCBPRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0287696-B1 ISOQUINOLINE DERIVATIVES Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1991-01-02 EP disclosed
US-4798897-A (AMINOALKYL)AMINOSULFONYL-SUBSTITUTED CARDIOVASCULAR AND RESPIRATORY SYSTEM DISORDERS ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1989-01-17 US disclosed
EP-0287696-A1 Isoquinoline derivatives Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1988-10-26 EP disclosed