SCHEMBL7326564

SCHEMBL7326564

O=S(=O)(c1cccc2cnccc12)N1CCC(O)C1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 11/20 0.65
ROCK1 Q13464 11/20 0.65
PRKD3 O94806 4/20 0.65
PRKCG P05129 4/20 0.65
PRKCB P05771 4/20 0.65
PRKCA P17252 4/20 0.65
PRKCH P24723 4/20 0.65
PRKCI P41743 4/20 0.65
PRKCE Q02156 4/20 0.65
PRKCQ Q04759 4/20 0.65
PRKCZ Q05513 4/20 0.65
PRKCD Q05655 4/20 0.65
PRKD1 Q15139 4/20 0.65
CYP3A4 P08684 3/20 0.65
CYP2D6 P10635 2/20 0.65
NFKB1 P19838 1/20 0.65
PRKACA P17612 3/20 0.62
PRKACG P22612 3/20 0.62
PRKACB P22694 3/20 0.62
ADORA3 P0DMS8 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7315524 0.93 CYP3A4 (0.62) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL7318375 0.93 ROCK2 (0.71) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL5083267 0.85 ROCK2 (0.68) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL23951500 0.85 PRKD3 (0.71) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL18477516 0.84 CYP3A4 (0.67) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL4727206 0.84 ROCK2 (0.66) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL4729640 0.82 ROCK2 (0.74) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL17228334 0.82 PRKD3 (0.65) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL4731780 0.82 ROCK2 (0.64) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL16712986 0.82 ROCK2 (0.61) ROCK2ROCK1PRKD3PRKCGPRKCB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0287696-B1 ISOQUINOLINE DERIVATIVES Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1991-01-02 EP disclosed
US-4798897-A (AMINOALKYL)AMINOSULFONYL-SUBSTITUTED CARDIOVASCULAR AND RESPIRATORY SYSTEM DISORDERS ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1989-01-17 US disclosed
EP-0287696-A1 Isoquinoline derivatives Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1988-10-26 EP disclosed