SCHEMBL7315714

SCHEMBL7315714

CCOC(=O)COC1CCN(C(=O)C(C)NC(=O)c2ccc(C(=N)NC(=O)c3ccccc3)cc2)CC1

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.75
ITGA2B P08514 10/20 0.75
KDM4E B2RXH2 1/20 0.41
PREP P48147 1/20 0.41
FAP Q12884 1/20 0.41
P2RY12 Q9H244 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM5 P08912 1/20 0.40
CHRM3 P20309 1/20 0.40
CCR1 P32246 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7308440 0.89 ITGB3 (0.70) ITGB3ITGA2BP2RY12CCR1
SCHEMBL7310770 0.86 ITGB3 (0.78) ITGB3ITGA2BCCR1
SCHEMBL7302533 0.85 ITGB3 (0.54) ITGB3ITGA2BKDM4EP2RY12CHRM2
Sibrafiban SCHEMBL27618015 0.81 ITGB3 (1.00) ITGB3ITGA2B
Sibrafiban SCHEMBL50759 0.81 ITGB3 (1.00) ITGB3ITGA2B
SCHEMBL13283231 0.78 ITGB3 (0.67) ITGB3ITGA2BPREPFAP
SCHEMBL7307129 0.77 ITGB3 (0.60) ITGB3ITGA2BKDM4EP2RY12CHRM2
Ro-44-3888 SCHEMBL7284509 0.76 ITGB3 (1.00) ITGB3ITGA2B
Ro-44-3888 SCHEMBL7283142 0.76 ITGB3 (1.00) ITGB3ITGA2B
SCHEMBL8770179 0.75 ITGB3 (0.74) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed