SCHEMBL7316169

SCHEMBL7316169

O=C(O)c1ccc(-n2ccc(=O)cc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.69
DDAH1 O94760 1/20 0.57
CA12 O43570 7/20 0.50
CA9 Q16790 7/20 0.50
CA1 P00915 6/20 0.50
ADH5 P11766 1/20 0.50
TP53 P04637 1/20 0.50
TSHR P16473 1/20 0.50
CA2 P00918 3/20 0.47
SCN2A Q99250 1/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
APEX1 P27695 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
NPSR1 Q6W5P4 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL217623 0.83 AOC2 (0.60) KMT2ADDAH1CA12CA9CA1
SCHEMBL334849 0.82 KMT2A (1.00) KMT2ATSHRALDH1A1MEN1MAPT
SCHEMBL1377974 0.82 KMT2A (0.67) KMT2ADDAH1CA1TSHRCA2
SCHEMBL7348821 0.82 KMT2A (0.67) KMT2ADDAH1ADH5ALDH1A1MEN1
SCHEMBL9595456 0.77 KMT2A (0.66) KMT2ATSHRKDM4EALDH1A1MEN1
SCHEMBL20649339 0.76 KMT2A (0.59) KMT2ACA12CA9CA1CA2
SCHEMBL7319404 0.75 KMT2A (0.52) KMT2AKDM4EALDH1A1MEN1POLB
SCHEMBL10195813 0.75 ADH5 (0.63) DDAH1ADH5TP53TSHR
SCHEMBL29171463 0.75 DDAH1 (0.47) KMT2ADDAH1CA12CA9CA1
SCHEMBL1664108 0.72 QPCT (0.58) KMT2ADDAH1CA12CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5783114-A PYRIMIDINE OR PYRIDAZINES MIXED WITH OTHER LIQUID CRYSTALLINE MATERIALS INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 1998-07-21 US disclosed
US-5246928-A Cardiovascular disorders SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-09-21 US disclosed
US-5066653-A Cardiovascular disorders; bronchodilators; phosphodiesterase inhibitors SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-19 US disclosed
CN-1009092-B The preparation method of Pyridione derivatives SMITH KLINE FRENCH LAB (GB) 1990-08-08 CN disclosed
US-4906628-A N-phenylpyridone type III phosphodiesterases SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1990-03-06 US disclosed
CN-86106546-A The preparation method of Pyridione derivatives 1987-05-20 CN disclosed
EP-0220044-A2 4(4-oxo-1,4-dihydropyridin-1-yl)phenyl derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1987-04-29 EP disclosed