SCHEMBL7316283

SCHEMBL7316283

C=CCN(Cc1ccc(Cl)cc1)C1CCC(=O)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 2/20 0.40
C5AR1 P21730 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
CYP2C19 P33261 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KDM4C Q9H3R0 1/20 0.35
BCL2A1 Q16548 5/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
KCNH2 Q12809 1/20 0.34
CHIT1 Q13231 1/20 0.34
CHIA Q9BZP6 1/20 0.34
DRD2 P14416 2/20 0.33
DRD3 P35462 2/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7319018 0.82 GRIN2B (0.47) LSSC5AR1CYP3A4CYP2D6CYP2C9
SCHEMBL1044449 0.78 SIGMAR1 (0.33) LSS
SCHEMBL7321429 0.75 HRH3 (0.50) LSSC5AR1CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL7313064 0.71 DRD2 (0.50) DRD2DRD3
SCHEMBL10320551 0.71 YTHDC1 (0.54) SLC6A2SLC6A4SLC6A3ALDH1A1RAB9A
SCHEMBL385070 0.71 YTHDC1 (0.54) SLC6A2SLC6A4SLC6A3ALDH1A1RAB9A
SCHEMBL24423760 0.68 DRD2 (0.47) ALDH1A1HTTDRD2DRD3CNR2
SCHEMBL7852342 0.68 HDAC3 (0.33) LSSSLC6A2SLC6A4
SCHEMBL7859419 0.66 ALDH1A1 (0.42) ALDH1A1HTTKCNH2DRD2LMNA
SCHEMBL6785682 0.65 ALDH1A1 (0.50) CYP3A4SLC6A2SLC6A4ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4886812-A REGULATING DOPAMINE CONCENTRATION; PARKINSON DISEASE, HYPOTENSIVE AGENT, SCHIZOPHRENIA DR. KARL THOMAE GMBH (DE) 1989-12-12 US disclosed
US-4843086-A HYPOTENSIVE AGENTS, SCHIZOPHRENIA, PARKINSON'S DISEASE BOEHRINGER INGELHEIM KG (DE) 1989-06-27 US disclosed
US-4731374-A PARKINSON*S DISEASE DR. KARL THOMAE GMBH (DE) 1988-03-15 US disclosed
EP-0186087-A1 Tetrahydro-benzothiazoles, their production and their use as intermediates or drugs Dr. Karl Thomae GmbH (DE) 1986-07-02 EP disclosed