SCHEMBL7318315

SCHEMBL7318315

S=C1CN=C(c2ccccc2Br)c2cc(Br)ccc2N1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 8/20 0.74
ALOX12 P18054 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
GABRA1 P14867 4/20 0.55
GABRA5 P31644 4/20 0.55
GABRA3 P34903 4/20 0.55
GABRA2 P47869 4/20 0.55
GABRB2 P47870 3/20 0.55
ALDH1A1 P00352 1/20 0.52
PKM P14618 1/20 0.52
HTT P42858 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
GABRG2 P18507 2/20 0.51
GABRB3 P28472 2/20 0.51
ADRA1A P35348 1/20 0.48
KMT2A Q03164 1/20 0.48
CCNB2 O95067 1/20 0.41
CDK1 P06493 1/20 0.41
CCNB1 P14635 1/20 0.41
GSK3B P49841 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11733821 0.87 CHRM1 (0.55) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL7324283 0.87 CHRM1 (0.73) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL11826679 0.87 ALOX12 (0.77) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL2843067 0.85 CHRM1 (1.00) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL18166494 0.84 GABRA1 (0.77) CHRM1GABRA1GABRA5GABRA3GABRA2
SCHEMBL7374778 0.81 ADRA1A (0.74) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL23881501 0.79 CHRM1 (0.67) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL30202099 0.79 CHRM1 (0.67) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL11828620 0.78 CHRM1 (0.65) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL18166492 0.75 GABRA1 (0.48) CHRM1GABRA1GABRA5GABRA3GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4902794-A Triazolo-benzodiazepines THE UPJOHN COMPANY (US) 1990-02-20 US disclosed
US-3987052-A SEDATIVES, TRANQUILIZERS, MUSCLE RELAXANTS THE UPJOHN COMPANY (US) 1976-10-19 US disclosed