SCHEMBL7319786

SCHEMBL7319786

CC(=O)N(C)c1ccc(C[C@H](NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(C)cc2)C(=O)OC(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 3/20 0.54
ITGB1 P05556 5/20 0.46
ITGA5 P08648 3/20 0.46
L3MBTL1 Q9Y468 3/20 0.45
MAPK1 P28482 2/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
ALDH1A1 P00352 1/20 0.45
FKBP1A P62942 1/20 0.45
MAPT P10636 2/20 0.44
TSHR P16473 2/20 0.44
RAB9A P51151 1/20 0.44
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.43
ITGAV P06756 1/20 0.43
ITGB7 P26010 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7321266 0.89 ITGA4 (0.61) ITGA4ITGB1ITGA5L3MBTL1MAPK1
SCHEMBL7066750 0.87 FKBP1A (0.58) ITGA4ITGB1ITGA5L3MBTL1MAPK1
SCHEMBL6708385 0.87 KMT2A (0.56) ITGA4ITGB1ITGA5L3MBTL1MAPK1
SCHEMBL3851005 0.86 ITGA4 (0.53) ITGA4ITGB1ITGA5L3MBTL1MAPK1
SCHEMBL7327448 0.85 ITGA4 (0.54) ITGA4ITGB1ITGA5L3MBTL1MAPK1
SCHEMBL3855551 0.84 ITGA4 (0.54) ITGA4ITGB1ITGA5L3MBTL1MAPK1
SCHEMBL3850548 0.83 ITGA4 (0.50) ITGA4ITGB1ITGA5MAPK1GAA
SCHEMBL6633729 0.83 ITGA4 (0.52) ITGA4ITGB1ITGA5L3MBTL1MAPK1
SCHEMBL6712256 0.82 ITGA4 (0.52) ITGA4ITGB1ITGA5L3MBTL1MAPK1
SCHEMBL7180720 0.82 ITGA4 (0.54) ITGA4ITGB1ITGA5L3MBTL1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001972-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP claimed
WO-1999006431-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed
US-6492421-B1 BINDING VERY LATE ANTIGEN-4; INFLAMMATORY DISEASES SUCH AS ASTHMA, ALZHEIMER'S DISEASE, ATHEROSCLEROSIS, AIDS, DEMENTIA, DIABETES, INFLAMMATORY BOWEL DISEASE, RHEUMATOID ARTHRITIS, TISSUE TRANSPLANTATION, TUMOR METASTASIS, MYOCARDIAL ISCHEMIA ATHENA NEUROSCIENCES, INC. 2002-12-10 US disclosed