SCHEMBL7319817

SCHEMBL7319817

COc1ccc2c(c1OC)CC(c1ccccc1)C1=C2CN(Cc2ccccc2)C1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44
ACHE P22303 5/20 0.39
BACE1 P56817 4/20 0.39
BCHE P06276 3/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
P4HB P07237 1/20 0.38
RAB9A P51151 1/20 0.38
PAX8 Q06710 1/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
SLC6A12 P48065 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9802089 0.88 SIGMAR1 (0.44) MEN1KMT2ANPC1P4HBRAB9A
SCHEMBL7439704 0.78 CYP2D6 (0.41) DRD2DRD3ACHEKMT2A
SCHEMBL8829448 0.76 ACHE (0.39) DRD2DRD4DRD3ACHE
Hydrochloric Acid SCHEMBL7307142 0.74 ACHE (0.41) ACHENPC1RAB9A
SCHEMBL8829332 0.73 ACHE (0.40) ACHEMEN1KMT2A
SCHEMBL6384149 0.67 BCHE (0.68) DRD4ACHEBACE1BCHE
Hydrochloric Acid SCHEMBL10828111 0.65 DRD2 (0.49) DRD2DRD3ACHEBACE1BCHE
SCHEMBL7313225 0.64 ALDH1A1 (0.55) ACHEMEN1KMT2ANPC1RAB9A
Hydrochloric Acid SCHEMBL7502831 0.64 ACHE (0.38) ACHE
Hydrochloric Acid SCHEMBL11262602 0.64 BCHE (0.50) DRD2ACHEBACE1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5621133-A PREPARING A 1-(3,4-DIALKOXYPHENYL),3-HYDROXYALKANE(C6-C12) BY EPOXIDIZING A HALO DERIVATIVE WITH A BASE FOLLOWED BY DECYCLICIZING WITH AN ORGANOMETALLIC COMPOUND IN A SOLVENT; NAPHTHYLENES, ISOCHROMENES AND ISOTHIOCHROMENES DENINNO MICHAEL P (US) 1997-04-15 US disclosed
US-5591884-A PROTECTED HYDROXYALKYLCATECHOL INTERMEDIATES ABBOTT LABORATORIES (US) 1997-01-07 US disclosed
WO-1996038435-A1 DOPAMINE AGONISTS ABBOTT LABORATORIES (US) 1996-12-05 WO disclosed
EP-0474767-B1 DOPAMINE AGONISTS ABBOTT LAB (US) 1996-02-21 EP disclosed
EP-0474767-A4 DOPAMINE AGONISTS 1992-07-08 EP disclosed
EP-0474767-A1 DOPAMINE AGONISTS. ABBOTT LAB (US) 1992-03-18 EP disclosed
WO-1990015056-A1 DOPAMINE AGONISTS ABBOTT LABORATORIES (US) 1990-12-13 WO disclosed
US-4963568-A TREATMENT OF PARKINSON*S DISEASE, CARDIOVASCULAR DISORDERS ABBOTT LABORATORIES (US) 1990-10-16 US disclosed