SCHEMBL7320052

SCHEMBL7320052

Nc1ccc(C(=O)NCO)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.71
MAPT P10636 1/20 0.71
HIF1A Q16665 1/20 0.71
SLC22A6 Q4U2R8 1/20 0.71
SLC22A8 Q8TCC7 1/20 0.71
LMNA P02545 3/20 0.55
MEN1 O00255 1/20 0.55
POLB P06746 1/20 0.55
PKM P14618 1/20 0.55
APEX1 P27695 1/20 0.55
KMT2A Q03164 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
TSHR P16473 2/20 0.54
SLC22A2 O15244 1/20 0.54
SLC22A1 O15245 1/20 0.54
ALDH1A1 P00352 1/20 0.54
ACHE P22303 1/20 0.54
MAPK1 P28482 1/20 0.54
CYP2C19 P33261 1/20 0.54
EPHX2 P34913 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4349764 0.89 THRB (0.55) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL9344489 0.84 KDM4E (0.68) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL853629 0.83 KDM4E (0.61) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL1913984 0.83 KDM4E (0.72) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL11132564 0.83 KDM4E (0.72) KDM4EMAPTHIF1ASLC22A6SLC22A8
Aminohippuric Acid SCHEMBL196513 0.83 KDM4E (1.00) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL10918143 0.83 EPHX2 (0.53) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL13113151 0.82 MAPT (0.70) KDM4EMAPTHIF1ASLC22A6SLC22A8
Aminohippuric Acid SCHEMBL31038605 0.82 KDM4E (0.96) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL11353059 0.81 KDM4E (0.63) KDM4EMAPTHIF1ASLC22A6SLC22A8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0271059-B1 2-Methylthiomethyl-dihydropyridines, a process for their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA (IT) 1993-10-20 EP disclosed
US-4971984-A Cardiovascular disorders, hypotensive agints BEEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1990-11-20 US disclosed
EP-0271059-A1 2-Methylthiomethyl-dihydropyridines, a process for their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1988-06-15 EP disclosed