SCHEMBL7322941

SCHEMBL7322941

CCOC(=O)OC1=C(C)NC(C)=C(OC(=O)OCC)C1c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.58
KDM4E B2RXH2 6/20 0.48
ALDH1A1 P00352 4/20 0.48
GAA P10253 2/20 0.48
TSHR P16473 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CACNA1D Q01668 2/20 0.47
CACNA1F O60840 1/20 0.47
CACNA1S Q13698 1/20 0.47
CACNA1C Q13936 1/20 0.47
ABCC1 P33527 1/20 0.47
DHFR P00374 1/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
LMNA P02545 1/20 0.46
CACNA1B Q00975 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CASP1 P29466 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10530880 0.92 ADORA3 (0.50) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL10786897 0.86 ADORA3 (0.52) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL11350249 0.86 ADORA3 (0.47) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL9369030 0.85 CACNA1F (0.49) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL11344156 0.84 ADORA3 (0.48) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL11005887 0.84 CACNA1B (0.49) ADORA3CACNA1DCACNA1FCACNA1SCACNA1C
SCHEMBL7298685 0.83 ADORA3 (0.45) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL9359378 0.83 ADORA3 (0.47) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL11329664 0.83 ADORA3 (0.47) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL9691613 0.82 ADORA3 (0.49) ADORA3KDM4EALDH1A1GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0288758-B1 DIHYDROPYRIDINAMIDES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN MEDICINES BAYER AG (DE) 1991-08-14 EP disclosed
EP-0229381-B1 METHIONINE-SUBSTITUTED 1,4-DIHYDROPYRIDINES, PROCESS FOR THE PREPARATION AND THEIR USE BAYER AG (DE) 1990-05-30 EP disclosed
EP-0362632-A2 Basic 4-aryl-DHP amides, process for their preparation and their pharmaceutical use BAYER AG (DE) 1990-04-11 EP disclosed
EP-0288758-A2 Dihydropyridinamides, process for their preparation and their use in medicines BAYER AG (DE) 1988-11-02 EP disclosed
EP-0236838-A2 Aminoester-dihydropyridines, process for their preparation and their use BAYER AG (DE) 1987-09-16 EP disclosed
EP-0229381-A1 Methionine-substituted 1,4-dihydropyridines, process for the preparation and their use BAYER AG (DE) 1987-07-22 EP disclosed
EP-0218068-A1 Dihydropyridine-2-hydroxyamines, process for their preparation and their use in medicaments BAYER AG (DE) 1987-04-15 EP disclosed
EP-0110259-B1 1,4-DIHYDROPYRIDINES, PROCESSES FOR THEIR PREPARATION AND THEIR USE IN MEDICINES BAYER AG (DE) 1986-12-17 EP disclosed
EP-0199238-A1 1,4-Dihydropyridine derivatives, process for their preparation and their use in medicaments BAYER AG (DE) 1986-10-29 EP disclosed
EP-0088274-B1 1,4-DIHYDROPYRIDINES, PROCESS FOR THEIR PREPARATION AND THEIR APPLICATION AS PHARMACEUTICAL PREPARATIONS BAYER AG (DE) 1986-09-03 EP disclosed
EP-0179386-A2 1,4-Dihydropyridine hydroxyamines, process for their preparation and their use as pharmaceutical agents BAYER AG (DE) 1986-04-30 EP disclosed
EP-0088276-B1 COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICAL PREPARATIONS BAYER AG (DE) 1986-04-30 EP disclosed
EP-0110259-A1 1,4-Dihydropyridines, processes for their preparation and their use in medicines BAYER AG (DE) 1984-06-13 EP disclosed
EP-0104550-A2 Condensed 1,4-dihydropyridines, process for their preparation and their application as pharmaceutical products BAYER AG (DE) 1984-04-04 EP disclosed
EP-0088276-A1 Compounds, process for their preparation and their use as pharmaceutical preparations BAYER AG (DE) 1983-09-14 EP disclosed
EP-0088274-A1 1,4-Dihydropyridines, process for their preparation and their application as pharmaceutical preparations BAYER AG (DE) 1983-09-14 EP disclosed
EP-0039863-A1 1,4-Dihydropyridines with different substituents in positions 2 and 6, processes for their preparation and their use in medicines BAYER AG (DE) 1981-11-18 EP disclosed