SCHEMBL7323669

SCHEMBL7323669

COc1c(C(=O)O)c2ccccc2n1CC1CCN(CCN(C(=O)OCc2ccccc2)S(C)(=O)=O)CC1.COc1c(C(=O)OCC2CCN(CCN(C(=O)OCc3ccccc3)S(C)(=O)=O)CC2)c2ccccc2n1C

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 9/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
NFKB1 P19838 1/20 0.39
PMP22 Q01453 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KCNH2 Q12809 5/20 0.38
AGTR1 P30556 1/20 0.38
ACHE P22303 2/20 0.36
BCHE P06276 1/20 0.36
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
CARM1 Q86X55 1/20 0.34
PRMT6 Q96LA8 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9704184 0.93 HTR4 (0.44) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7322685 0.85 CYP2C9 (0.51) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7340946 0.83 HTR4 (0.47) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7325668 0.83 OPRM1 (0.37) HTR4AGTR1
SCHEMBL7301885 0.74 HTR4 (0.67) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7300816 0.73 HTR4 (0.54) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL16504002 0.66 CYP2C9 (0.66) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7302781 0.65 HTR4 (0.45) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7301907 0.65 CYP2C9 (0.53) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7304670 0.64 KDM1A (0.46) AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP disclosed
WO-1992014727-A1 3-PIPERIDINYLMETHYLCARBOXYLATE SUBSTITUTED INDOLES GLAXO GROUP LIMITED (GB) 1992-09-03 WO disclosed
EP-0501322-A1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LIMITED (GB) 1992-09-02 EP disclosed