SCHEMBL7323916

SCHEMBL7323916

O=C1Cc2ccc3ccccc3c2NN1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 1/20 0.41
PAX8 Q06710 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
HSD17B10 Q99714 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2A6 P11509 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
AHR P35869 2/20 0.36
PDK2 Q15119 1/20 0.36
PARP1 P09874 1/20 0.36
LMNA P02545 1/20 0.36
HPRT1 P00492 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2905322 0.84 AHR (0.49) ANPEPPAX8CA12CA1CA2
SCHEMBL1159910 0.72 ALDH1A1 (0.42) ANPEPPAX8CA12CA1CA2
SCHEMBL28986962 0.71 NPC1 (0.59) CA9HSD17B10AHRPDK2
SCHEMBL6722121 0.71 NPC1 (0.47) PAX8CA12CA1CA2CA4
SCHEMBL636014 0.70 TDP2 (0.51) ANPEPAHRPDK2
SCHEMBL12799615 0.69 HSD17B10 (0.39) ANPEPCA12CA1CA2CA4
SCHEMBL10723285 0.69 ALDH1A1 (0.39) ANPEPCA12CA1CA2CA4
SCHEMBL16254014 0.68 HSD17B10 (0.46) PAX8CA12CA1CA2CA4
SCHEMBL29616441 0.68 HSD17B10 (0.46) PAX8CA12CA1CA2CA4
SCHEMBL21196716 0.68 NPC1 (0.44) ANPEPCA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5246928-A Cardiovascular disorders SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-09-21 US disclosed
US-5066653-A Cardiovascular disorders; bronchodilators; phosphodiesterase inhibitors SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-19 US disclosed
US-4906628-A N-phenylpyridone type III phosphodiesterases SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1990-03-06 US disclosed
EP-0220044-A2 4(4-oxo-1,4-dihydropyridin-1-yl)phenyl derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1987-04-29 EP disclosed