SCHEMBL7324919

SCHEMBL7324919

CC(CO)C([C]=O)NC(=O)CCCC[C@@H](Cc1ccccc1)NC(=O)[C@H](C)N(C(=O)OCc1ccccc1)C(=O)[C@H](C)N

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.35
MAPK1 P28482 1/20 0.35
SIRT2 Q8IXJ6 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
CTSL P07711 2/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CTSK P43235 1/20 0.33
LPAR1 Q92633 2/20 0.33
LPAR3 Q9UBY5 2/20 0.33
MMP8 P22894 1/20 0.33
MMP14 P50281 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7329705 0.86 CTSD (0.40) CYP3A4MAPK1
SCHEMBL7324603 0.85 CTSD (0.42) CTSK
SCHEMBL7332055 0.83 CTSD (0.39)
SCHEMBL7330377 0.82 CTRB1 (0.43) CYP3A4SIRT2CYP1A2CYP2D6CYP2C9
SCHEMBL7324038 0.76 CTSD (0.40) CYP3A4MAPK1
SCHEMBL9295742 0.75 CYP3A4 (0.35) CYP3A4MAPK1CYP1A2CYP2D6CYP2C9
SCHEMBL10954138 0.72 ACE (0.45)
SCHEMBL7319644 0.70 CTSD (0.49)
SCHEMBL7328959 0.70 CTSD (0.49)
SCHEMBL7607048 0.70 ABCB1 (0.41) CTSLALDH1A1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1990000399-A1 RETROVIRAL PROTEASE BINDING PEPTIDES SMITHKLINE BECKMAN CORPORATION (US) 1990-01-25 WO disclosed
EP-0352000-A2 Retroviral protease binding peptides SMITHKLINE BEECHAM CORPORATION (US) 1990-01-24 EP disclosed