SCHEMBL7325202

SCHEMBL7325202

NCCCNCCCN(CCCN)C(=O)Cc1ccccc1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.49
MC3R P41968 6/20 0.47
MC4R P32245 5/20 0.47
MC5R P33032 4/20 0.47
CA12 O43570 5/20 0.43
CA2 P00918 5/20 0.43
CA9 Q16790 5/20 0.43
CA1 P00915 1/20 0.43
CA3 P07451 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
KDM4E B2RXH2 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
AKR1B1 P15121 1/20 0.41
MPO P05164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7328587 0.83 CYP3A4 (0.59) TSHR
SCHEMBL7320232 0.78 REN (0.55) RENMC3RMC4R
SCHEMBL7327795 0.77 REN (0.53) RENMC3RMC4RMC5R
SCHEMBL7321088 0.76 CA12 (0.70) CA12CA2CA9CA1CA3
SCHEMBL21498143 0.73 REN (0.55) RENMC3RMC4RMC5R
SCHEMBL7319791 0.72 REN (0.50) RENMC3RMC4RKDM4E
SCHEMBL9098622 0.72 CA12 (0.79) CA12CA2CA9KDM4ETSHR
SCHEMBL26087539 0.71 CA12 (0.77) CA12CA2CA9KDM4ETSHR
SCHEMBL18096448 0.71 CA12 (0.77) CA12CA2CA9KDM4ETSHR
SCHEMBL22566158 0.70 MC3R (0.58) RENMC3RMC4RMC5RCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5218000-A Nervous system disorders, antiischemic agents NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1993-06-08 US disclosed
EP-0361687-A1 Therapeutic polyamine-amides BTG INTERNATIONAL LIMITED (GB) 1990-04-04 EP disclosed
WO-1990002114-A1 THERAPEUTIC POLYAMINE-AMIDES NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1990-03-08 WO disclosed