SCHEMBL7328587

SCHEMBL7328587

COc1ccccc1CC(=O)N(CCCN)CCCNCCCN

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.59
CYP2D6 P10635 2/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2C19 P33261 1/20 0.59
TSHR P16473 2/20 0.56
ACHE P22303 6/20 0.55
CHRM2 P08172 11/20 0.53
BCHE P06276 5/20 0.47
TOP2A P11388 2/20 0.47
GRIN1 Q05586 4/20 0.46
GRIN2A Q12879 4/20 0.46
TP53 P04637 1/20 0.46
CHRM4 P08173 1/20 0.46
CHRM5 P08912 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
THPO P40225 1/20 0.46
RECQL P46063 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7325202 0.83 REN (0.49) TSHR
SCHEMBL7319791 0.78 REN (0.50) CHRM2
SCHEMBL9447512 0.78 CA12 (0.65) CYP3A4CYP2D6TSHRACHECHRM2
SCHEMBL10013764 0.73 CYP1A2 (0.78) CYP3A4CYP2D6CYP1A2CYP2C19TSHR
SCHEMBL10873043 0.73 CHRM2 (0.85) CYP3A4CYP2D6TSHRACHECHRM2
SCHEMBL25695874 0.72 CDK8 (0.49)
SCHEMBL7320232 0.72 REN (0.55) GRIN1GRIN2A
SCHEMBL7327795 0.71 REN (0.53)
SCHEMBL21498147 0.71 ELANE (0.52) CYP3A4CYP1A2CYP2C19TSHR
SCHEMBL8567854 0.70 TSHR (0.60) CYP3A4CYP2D6CYP1A2CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5218000-A Nervous system disorders, antiischemic agents NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1993-06-08 US disclosed
EP-0361687-A1 Therapeutic polyamine-amides BTG INTERNATIONAL LIMITED (GB) 1990-04-04 EP disclosed
WO-1990002114-A1 THERAPEUTIC POLYAMINE-AMIDES NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1990-03-08 WO disclosed