SCHEMBL7325866

SCHEMBL7325866

CC1(C)Oc2ccc(C#N)cc2C(Nc2ccc(O)nn2)C1(C)O

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 8/20 0.39
ABCC9 O60706 7/20 0.39
KDM4E B2RXH2 1/20 0.38
KCNE1 P15382 2/20 0.36
KCNQ1 P51787 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7335715 0.84 ALDH1A1 (0.30)
SCHEMBL7330716 0.82 ABCB1 (0.41) ABCB1ABCC9KDM4E
SCHEMBL7358720 0.81 ABCC9 (0.41) ABCB1ABCC9KDM4EKCNE1KCNQ1
SCHEMBL7330935 0.80 ABCB1 (0.39) ABCB1ABCC9KDM4E
SCHEMBL8541387 0.80 ABCB1 (0.40) ABCB1ABCC9KDM4E
SCHEMBL8539388 0.80 ABCB1 (0.40) ABCB1ABCC9KDM4E
SCHEMBL8544061 0.80 ABCB1 (0.40) ABCB1ABCC9KDM4E
SCHEMBL7330928 0.80 ABCC9 (0.56) ABCB1ABCC9
SCHEMBL7273801 0.79 ABCC9 (0.39) ABCB1ABCC9KDM4E
SCHEMBL7331870 0.77 ABCC9 (0.39) ABCB1ABCC9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0363883-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1990-04-18 EP disclosed