SCHEMBL7326496

SCHEMBL7326496

NCCc1c[nH]c2ccc(-c3ccccn3)cc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 6/20 0.57
HTR1B P28222 5/20 0.57
HTR1A P08908 7/20 0.55
HTR2A P28223 7/20 0.55
HTR2C P28335 5/20 0.55
MPO P05164 2/20 0.55
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2D6 P10635 2/20 0.55
HTR7 P34969 2/20 0.55
HTR6 P50406 2/20 0.55
TAAR1 Q96RJ0 2/20 0.55
CYP2A6 P11509 1/20 0.55
NFKB1 P19838 1/20 0.55
CTSK P43235 1/20 0.55
CYP2A13 Q16696 1/20 0.55
LTA4H P09960 1/20 0.54
PLA2G2A P14555 1/20 0.54
PMP22 Q01453 1/20 0.54
TRPM8 Q7Z2W7 5/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7331855 0.83 HTR1D (0.60) HTR1DHTR1BHTR1AHTR2AHTR2C
SCHEMBL2536567 0.81 LTA4H (0.67) HTR1DHTR1BHTR1AHTR2AHTR2C
SCHEMBL7359803 0.80 CSNK2A1 (0.55) MPOCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8475787 0.78 HTR1D (0.54) HTR1DHTR1BHTR1AHTR2AHTR2C
SCHEMBL31370163 0.77 KMT2A (0.62) HTR1AHTR2AHTR2CMPOCYP3A4
Hydrochloric Acid SCHEMBL7313598 0.77 LTA4H (0.65) HTR1DHTR1BHTR1AHTR2AHTR2C
Hydrochloric Acid SCHEMBL9238831 0.76 HTR6 (0.58) HTR1DHTR1BHTR1AHTR2AHTR2C
SCHEMBL7334745 0.75 HTR1D (0.64) HTR1DHTR1BHTR1AHTR2AHTR2C
SCHEMBL8869386 0.75 TRPM8 (0.70) HTR1DHTR1BHTR1AHTR2AHTR2C
SCHEMBL7325860 0.75 LTA4H (0.59) HTR1DHTR1BHTR1AHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674620-A1 TRYPTAMINE ANALOGUES AS 5-HT 1?-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-10-04 EP claimed
WO-1994014771-A1 TRYPTAMINE ANALOGUES AS 5-HT1-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO claimed
EP-0674620-A1 TRYPTAMINE ANALOGUES AS 5-HT 1?-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-10-04 EP disclosed
WO-1994014771-A1 TRYPTAMINE ANALOGUES AS 5-HT1-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO disclosed