SCHEMBL7328255

SCHEMBL7328255

COc1ccc(-c2ccc3[nH]cc(C4=CCNC(C)C4)c3c2)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.47
MAP3K11 Q16584 1/20 0.45
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
HTR1D P28221 1/20 0.41
HTR2C P28335 1/20 0.41
MAPK1 P28482 1/20 0.41
BRCA1 P38398 1/20 0.41
HTR6 P50406 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PRKAG1 P54619 1/20 0.40
PRKAA1 Q13131 1/20 0.40
PRKAB1 Q9Y478 1/20 0.40
PIM2 Q9P1W9 2/20 0.39
JAK2 O60674 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7327374 0.76 SLC6A4 (0.65)
SCHEMBL6625901 0.74 HTR2C (0.41) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL7205820 0.74 SLC6A4 (0.53) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL2522333 0.73 MAP3K11 (0.80) TDO2MAP3K11CYP3A4MAPK1PRKAG1
SCHEMBL6841621 0.69 HTR1D (0.49) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL6497949 0.69 TDO2 (0.46) TDO2
SCHEMBL3627714 0.66 CDK7 (0.38) TDO2KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL16192164 0.66 TYK2 (0.70) MAP3K11PIM2PIM1PIM3
SCHEMBL18136456 0.65 DYRK1A (0.49) MAP3K11CYP3A4HTR2CJAK2PRKD3
SCHEMBL18129649 0.65 DYRK1A (0.49) MAP3K11CYP3A4HTR2CJAK2PRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674620-A1 TRYPTAMINE ANALOGUES AS 5-HT 1?-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-10-04 EP claimed
WO-1994014771-A1 TRYPTAMINE ANALOGUES AS 5-HT1-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO claimed