SCHEMBL6625901

SCHEMBL6625901

CC1CC(c2c[nH]c3ccc(O)cc23)=CCN1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.41
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HTR6 P50406 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 2/20 0.41
HTR1D P28221 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
BRCA1 P38398 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2D6 P10635 3/20 0.41
THPO P40225 1/20 0.41
NFKB1 P19838 2/20 0.40
LMNA P02545 1/20 0.40
GLA P06280 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7205820 0.84 SLC6A4 (0.53) HTR2CCYP1A2CYP3A4ALDH1A1HTR6
SCHEMBL6841621 0.77 HTR1D (0.49) HTR2CCYP1A2CYP3A4ALDH1A1HTR6
SCHEMBL6497949 0.76 TDO2 (0.46) SLC6A4
SCHEMBL3836149 0.75 HTR6 (0.67) HTR2CCYP1A2CYP3A4ALDH1A1HTR6
SCHEMBL5435851 0.74 HTR2C (0.56) HTR2CCYP1A2CYP3A4ALDH1A1HTR6
SCHEMBL7328255 0.74 TDO2 (0.47) HTR2CCYP1A2CYP3A4ALDH1A1HTR6
SCHEMBL8798676 0.73 HTR2B (0.40) HTR2CALDH1A1HTR6KDM4EMEN1
SCHEMBL5367487 0.69 SLC6A4 (0.76) HTR6KDM4EHSD17B10LMNAHTR1A
SCHEMBL6492415 0.69 AR (0.42) HTR1DHTR2A
SCHEMBL13302269 0.68 DYRK1A (0.55) HTR2CCYP1A2CYP3A4ALDH1A1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377580-A2 BENZENESULFONIC ACID INDOL-5-YL ESTERS AS ANTAGONISTS OF THE 5-HT6 RECEPTOR ELI LILLY AND COMPANY (US) 2004-01-07 EP disclosed
WO-2002060871-A2 BENZENESULFONIC ACID INDOL-5-YL ESTERS AS ANTAGONISTS OF THE 5-HT6 RECEPTOR ELI LILLY AND COMPANY (US) 2002-08-08 WO disclosed