SCHEMBL7328822

SCHEMBL7328822

CCCN(c1cccc(OCC(=O)O)c1)S(=O)(=O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.54
CA12 O43570 3/20 0.49
CA1 P00915 3/20 0.49
CA2 P00918 3/20 0.49
CA4 P22748 3/20 0.49
CA9 Q16790 3/20 0.49
PSEN1 P49768 1/20 0.48
PSEN2 P49810 1/20 0.48
APH1B Q8WW43 1/20 0.48
NCSTN Q92542 1/20 0.48
APH1A Q96BI3 1/20 0.48
PSENEN Q9NZ42 1/20 0.48
MAPT P10636 3/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
LMNA P02545 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7335466 0.90 ESR1 (0.59) ESR1CA12CA1CA2CA4
SCHEMBL7324331 0.84 CA12 (0.61) ESR1CA12CA1CA2CA4
SCHEMBL8542191 0.83 F2 (0.60) CA12CA1CA2CA4CA9
SCHEMBL7334512 0.82 ESR1 (0.55) ESR1CA12CA1CA2CA4
SCHEMBL7327551 0.79 ESR1 (0.55) ESR1MAPTGAANPSR1LMNA
SCHEMBL7327957 0.78 MEN1 (0.58) CA12CA1CA2CA4CA9
SCHEMBL10438567 0.77 ESR1 (0.79) ESR1LMNAL3MBTL1NR1I2KMT2A
SCHEMBL7333708 0.77 MAPT (0.60) CA12CA1CA2CA4CA9
SCHEMBL14878119 0.76 NR1I2 (0.57) ESR1MAPTGAALMNAKEAP1
SCHEMBL14878166 0.76 KEAP1 (0.49) ESR1MAPTGAALMNAKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687253-B1 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1998-12-16 EP disclosed
EP-0687253-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME Roche Diagnostics GmbH (DE) 1995-12-20 EP disclosed
WO-1994020467-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1994-09-15 WO disclosed