SCHEMBL7324331

SCHEMBL7324331

O=C(O)COc1cccc(N(Cc2ccccc2)S(=O)(=O)c2ccccc2)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 6/20 0.61
CA1 P00915 6/20 0.61
CA2 P00918 6/20 0.61
CA4 P22748 6/20 0.61
CA9 Q16790 6/20 0.61
MAPT P10636 5/20 0.60
LMNA P02545 3/20 0.60
NR3C1 P04150 1/20 0.57
ALDH1A1 P00352 1/20 0.57
ESR1 P03372 1/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
PTGES O14684 2/20 0.53
TP53 P04637 1/20 0.53
THRB P10828 1/20 0.53
PGR P06401 2/20 0.52
ALOX5 P09917 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7333708 0.87 MAPT (0.60) CA12CA1CA2CA4CA9
SCHEMBL7335466 0.86 ESR1 (0.59) CA12CA1CA2CA4CA9
SCHEMBL7328822 0.84 ESR1 (0.54) CA12CA1CA2CA4CA9
SCHEMBL7334512 0.83 ESR1 (0.55) CA12CA1CA2CA4CA9
SCHEMBL8547733 0.82 MAPT (0.71) MAPTLMNANR3C1MEN1KMT2A
SCHEMBL8542191 0.81 F2 (0.60) CA12CA1CA2CA4CA9
SCHEMBL214282 0.80 CRHBP (0.55) CA12CA1CA2CA4CA9
SCHEMBL7332305 0.80 PGR (0.55) CA12CA1CA2CA4CA9
SCHEMBL2189346 0.78 LMNA (0.85) MAPTLMNAALDH1A1ESR1MEN1
SCHEMBL6295954 0.78 ESR1 (0.71) MAPTLMNANR3C1ALDH1A1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687253-B1 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1998-12-16 EP disclosed
EP-0687253-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME Roche Diagnostics GmbH (DE) 1995-12-20 EP disclosed
WO-1994020467-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1994-09-15 WO disclosed