SCHEMBL7329537

SCHEMBL7329537

Cn1cc[n+]2cc(-c3ccc(Cl)cc3)[nH]c(=O)c12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.37
KDM4E B2RXH2 8/20 0.37
GAA P10253 5/20 0.37
THRB P10828 2/20 0.37
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
PARP1 P09874 2/20 0.35
HPGD P15428 4/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
PRKDC P78527 1/20 0.33
LMNA P02545 1/20 0.33
GLA P06280 1/20 0.33
CRHBP P24387 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337599 0.83 TNKS (0.39) ALDH1A1KDM4EPARP1TNKSTNKS2
SCHEMBL7328415 0.82 MAPT (0.38) ALDH1A1KDM4EGAAMAPTPARP1
SCHEMBL7331334 0.74 BRD4 (0.36) ALDH1A1KDM4EGAAMAPTTSHR
SCHEMBL7338197 0.73 CTSV (0.35) ALDH1A1KDM4EGAAMAPTPARP1
SCHEMBL7329545 0.69 TNKS (0.41) ALDH1A1KDM4EGAATHRBMAPT
SCHEMBL16664837 0.67 ALDH1A1 (0.51) ALDH1A1KDM4EGAATHRBMAPT
SCHEMBL19501571 0.59 MAPT (0.41) ALDH1A1KDM4EMAPTHPGDCYP2C9
SCHEMBL3918612 0.58 ALDH1A1 (0.51) ALDH1A1KDM4EGAATHRBMAPT
SCHEMBL7729347 0.58 KDM4E (0.52) ALDH1A1KDM4EGAATHRBMAPT
SCHEMBL7336678 0.57 TNKS (0.74) ALDH1A1KDM4EGAAMAPTPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726900-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS Aventis Pharma S.A. (FR) 1996-08-21 EP disclosed
WO-1995012594-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1995-05-11 WO disclosed