SCHEMBL7337599

SCHEMBL7337599

Cn1cc[n+]2cc(-c3ccc(C(F)(F)F)cc3)[nH]c(=O)c12

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TNKS O95271 5/20 0.39
PARP1 P09874 3/20 0.39
TDP2 O95551 1/20 0.34
PDE2A O00408 1/20 0.34
DAO P14920 1/20 0.34
COMT P21964 1/20 0.34
TNKS2 Q9H2K2 3/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ATM Q13315 1/20 0.33
PARP2 Q9UGN5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7329537 0.83 ALDH1A1 (0.37) TNKSPARP1TNKS2KDM4EALDH1A1
SCHEMBL7328415 0.79 MAPT (0.38) TNKSPARP1TNKS2KDM4EALDH1A1
SCHEMBL7337601 0.72 TNKS (0.43) TNKSPARP1COMTTNKS2PARP2
SCHEMBL7331334 0.71 BRD4 (0.36) PARP1TDP2KDM4EALDH1A1
SCHEMBL7338197 0.70 CTSV (0.35) PARP1KDM4EALDH1A1
SCHEMBL7397534 0.69 TNKS (0.41) TNKSPARP1TNKS2KDM4EALDH1A1
SCHEMBL15693150 0.68 TNKS (0.52) TNKSPARP1TNKS2KDM4EALDH1A1
SCHEMBL15614396 0.62 ERCC1 (0.67) TNKSPARP1COMTTNKS2
SCHEMBL15287390 0.62 TNKS (0.71) TNKSPARP1TNKS2PARP2
SCHEMBL15775516 0.61 TNKS (0.56) TNKSPARP1TNKS2ALDH1A1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726900-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS Aventis Pharma S.A. (FR) 1996-08-21 EP disclosed
WO-1995012594-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1995-05-11 WO disclosed