SCHEMBL7329545

SCHEMBL7329545

C[n+]1ccn2cc(-c3ccc(Cl)cc3)[nH]c(=O)c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 7/20 0.41
PARP1 P09874 5/20 0.41
TNKS2 Q9H2K2 5/20 0.41
ALDH1A1 P00352 7/20 0.40
GAA P10253 4/20 0.40
KDM4E B2RXH2 6/20 0.37
MAPT P10636 3/20 0.37
THRB P10828 2/20 0.37
TSHR P16473 1/20 0.37
RXFP1 Q9HBX9 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HPGD P15428 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
GLA P06280 1/20 0.33
CRHBP P24387 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7327605 0.87 TNKS (0.53) TNKSPARP1TNKS2ALDH1A1GAA
SCHEMBL7330451 0.84 BRD4 (0.41) TNKSPARP1TNKS2ALDH1A1GAA
SCHEMBL7336871 0.84 MAP2K1 (0.44) TNKSPARP1TNKS2ALDH1A1GAA
SCHEMBL7337601 0.83 TNKS (0.43) TNKSPARP1TNKS2
SCHEMBL7328423 0.82 MAPT (0.42) TNKSPARP1TNKS2ALDH1A1GAA
SCHEMBL7337908 0.80 SCN10A (0.38) TNKSPARP1TNKS2ALDH1A1GAA
SCHEMBL7328378 0.77 TNKS (0.38) TNKSPARP1TNKS2ALDH1A1KDM4E
SCHEMBL7336678 0.69 TNKS (0.74) TNKSPARP1TNKS2ALDH1A1GAA
SCHEMBL7397534 0.67 TNKS (0.41) TNKSPARP1TNKS2ALDH1A1KDM4E
SCHEMBL14469279 0.66 EGFR (0.41) PARP1ALDH1A1SMN1; SMN2HPGDCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726900-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS Aventis Pharma S.A. (FR) 1996-08-21 EP disclosed
WO-1995012594-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1995-05-11 WO disclosed