SCHEMBL7329617

SCHEMBL7329617

CCc1nc(Cl)c(Oc2cc(OC)ccc2Cl)c(Cl)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
GFER P55789 1/20 0.40
SLC6A4 P31645 5/20 0.40
HTR2A P28223 4/20 0.40
KCNH2 Q12809 3/20 0.40
KDM4E B2RXH2 1/20 0.40
DHPS P49366 3/20 0.38
EDNRA P25101 3/20 0.37
EDNRB P24530 2/20 0.37
GAA P10253 1/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
THRB P10828 1/20 0.34
SLC6A2 P23975 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328086 0.87 ALDH1A1 (0.40) ALDH1A1GFERSLC6A4HTR2AKCNH2
SCHEMBL8323583 0.85 ALDH1A1 (0.38) ALDH1A1GFERSLC6A4HTR2AKCNH2
SCHEMBL7298739 0.84 CDK1 (0.43) ALDH1A1GFERSLC6A4HTR2AKCNH2
SCHEMBL4435549 0.79 EDNRB (0.44) ALDH1A1SLC6A4HTR2AKCNH2KDM4E
SCHEMBL8323581 0.78 HTR2A (0.40) ALDH1A1GFERSLC6A4HTR2AKCNH2
SCHEMBL7330437 0.76 DHPS (0.59) ALDH1A1DHPSCA12CA1CA2
SCHEMBL7332509 0.76 RORC (0.38) ALDH1A1KDM4EGAA
SCHEMBL8328712 0.72 KMT2A (0.37) ALDH1A1SLC6A4HTR2AKCNH2KDM4E
SCHEMBL7417417 0.72 ALDH1A1 (0.47) ALDH1A1GFERKDM4EGAA
SCHEMBL858910 0.72 ALDH1A1 (0.50) ALDH1A1GFERKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526708-B1 Sulfonamide, preparation and use thereof as medicine and intermediate HOFFMANN LA ROCHE (CH) 2000-10-18 EP disclosed
US-5292740-A Sulfonamides HOFFMANN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0526708-A1 Sulfonamide, preparation and use thereof as medicine and intermediate F. HOFFMANN-LA ROCHE AG (CH) 1993-02-10 EP disclosed