SCHEMBL8323581

SCHEMBL8323581

COc1ccc(Cl)c(Oc2c(Cl)nc(C(C)OC)nc2Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.40
SLC6A4 P31645 4/20 0.40
KCNH2 Q12809 3/20 0.40
DHPS P49366 2/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
GAA P10253 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
P2RX3 P56373 1/20 0.34
P2RX2 Q9UBL9 1/20 0.34
ALDH1A1 P00352 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7298739 0.81 CDK1 (0.43) HTR2ASLC6A4KCNH2DHPSGAA
SCHEMBL7329617 0.78 ALDH1A1 (0.40) HTR2ASLC6A4KCNH2DHPSGAA
SCHEMBL4435549 0.77 EDNRB (0.44) HTR2ASLC6A4KCNH2GAAEDNRB
SCHEMBL8328086 0.77 ALDH1A1 (0.40) HTR2ASLC6A4KCNH2DHPSCYP11B1
SCHEMBL8323583 0.75 ALDH1A1 (0.38) HTR2ASLC6A4KCNH2DHPSGAA
SCHEMBL4427054 0.70 EDNRB (0.43) HTR2ASLC6A4KCNH2EDNRBEDNRA
SCHEMBL31179987 0.69 P2RX3 (0.52) HTR2ASLC6A4KCNH2DHPSGAA
SCHEMBL7009624 0.69 EDNRB (0.41) HTR2ASLC6A4KCNH2EDNRBEDNRA
SCHEMBL7010336 0.69 DHPS (0.41) DHPSEDNRBEDNRAALDH1A1HPGD
SCHEMBL8634388 0.69 HTR2A (0.36) HTR2ASLC6A4KCNH2DHPSGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0633259-B1 Sulfonylaminopyrimidines, their preparation and their use as medicine HOFFMANN LA ROCHE (CH) 1999-01-13 EP disclosed
US-5541186-A ENDOTHELIN RECEPTOR INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1996-07-30 US disclosed
EP-0633259-A1 Sulfonylaminopyrimidines, their preparation and their use as medicine F. HOFFMANN-LA ROCHE AG (CH) 1995-01-11 EP disclosed