SCHEMBL7330508

SCHEMBL7330508

NC(=O)NC(=O)c1ccccc1OCC1CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.53
CNR1 P21554 1/20 0.53
CNR2 P34972 1/20 0.53
MRGPRX1 Q96LB2 1/20 0.49
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 1/20 0.44
PARP15 Q460N3 1/20 0.43
PARP10 Q53GL7 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
SGMS2 Q8NHU3 2/20 0.43
SIRT2 Q8IXJ6 1/20 0.43
HCRTR1 O43613 1/20 0.42
CTSD P07339 1/20 0.42
RIPK1 Q13546 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4000543 0.83 ALDH1A1 (0.53) FAAHCNR1CNR2MRGPRX1MEN1
SCHEMBL17206382 0.81 FAAH (0.51) FAAHCNR1CNR2MRGPRX1PDE4A
SCHEMBL27854331 0.80 FAAH (0.51) FAAHCNR1CNR2MRGPRX1PDE4A
SCHEMBL933677 0.79 ALDH1A1 (0.57) FAAHCNR1CNR2MRGPRX1KMT2A
SCHEMBL11628242 0.77 RIPK1 (0.46) FAAHCNR1CNR2MRGPRX1PDE4A
SCHEMBL27983423 0.77 FAAH (0.52) FAAHCNR1CNR2MRGPRX1PDE4A
Hydrochloric Acid SCHEMBL7726218 0.76 HTR2C (0.48) FAAHCNR1CNR2MRGPRX1PDE4A
SCHEMBL7329125 0.76 FAAH (0.47) FAAHCNR1CNR2MRGPRX1MEN1
SCHEMBL1474965 0.74 IRAK4 (0.51) MEN1KMT2AALDH1A1PARP15PARP10
SCHEMBL11466965 0.74 PARP15 (0.49) FAAHCNR1CNR2MRGPRX1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422846-B1 Aroyl-ureas WYETH JOHN & BROTHER LTD (GB) 1994-02-16 EP claimed
EP-0422846-A2 Aroyl-ureas JOHN WYETH & BROTHER LIMITED (GB) 1991-04-17 EP claimed
US-5436251-A Treating neuro-psychiatric disorders gastrointenstinal disorders or migranes JOHN WYETH & BROTHER, LIMITED (GB) 1995-07-25 US disclosed
EP-0422846-B1 Aroyl-ureas WYETH JOHN & BROTHER LTD (GB) 1994-02-16 EP disclosed
EP-0422846-A2 Aroyl-ureas JOHN WYETH & BROTHER LIMITED (GB) 1991-04-17 EP disclosed