SCHEMBL27854331

SCHEMBL27854331

O=C(c1ccccc1OCC1CC1)c1ccccc1OCC1CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.51
CNR1 P21554 1/20 0.51
CNR2 P34972 1/20 0.51
MRGPRX1 Q96LB2 1/20 0.50
RIPK1 Q13546 1/20 0.49
HTR2C P28335 2/20 0.44
PARP15 Q460N3 1/20 0.44
PARP10 Q53GL7 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
PDE4A P27815 2/20 0.43
PDE4B Q07343 2/20 0.43
PDE4C Q08493 2/20 0.43
PDE4D Q08499 2/20 0.43
DRD2 P14416 1/20 0.42
DRD1 P21728 1/20 0.42
DRD3 P35462 1/20 0.42
ALDH1A1 P00352 2/20 0.42
KMT2A Q03164 2/20 0.42
ELANE P08246 1/20 0.42
PTK2B Q14289 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL933677 0.88 ALDH1A1 (0.57) FAAHCNR1CNR2MRGPRX1RIPK1
SCHEMBL27983423 0.86 FAAH (0.52) FAAHCNR1CNR2MRGPRX1RIPK1
SCHEMBL4000543 0.86 ALDH1A1 (0.53) FAAHCNR1CNR2MRGPRX1PARP15
SCHEMBL3064765 0.81 FAAH (0.54) FAAHCNR1CNR2MRGPRX1HTR2C
SCHEMBL29055574 0.81 FAAH (0.57) FAAHCNR1CNR2PARP15PARP10
SCHEMBL1388095 0.80 FAAH (0.60) FAAHCNR1CNR2PARP15PARP10
SCHEMBL9366238 0.80 FAAH (0.44) FAAHCNR1CNR2MRGPRX1RIPK1
SCHEMBL7330508 0.80 FAAH (0.53) FAAHCNR1CNR2MRGPRX1RIPK1
SCHEMBL11628242 0.79 RIPK1 (0.46) FAAHCNR1CNR2MRGPRX1RIPK1
SCHEMBL238499 0.79 PTGER1 (0.47) FAAHCNR1CNR2MRGPRX1RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102471314-B Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction ROTTAPHARM SPA 2015-05-13 CN claimed
CN-102471314-B Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction ROTTAPHARM SPA 2015-05-13 CN disclosed
CN-102471314-A Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction ROTTAPHARM SPA 2012-05-23 CN disclosed