SCHEMBL7334663

SCHEMBL7334663

CC1(C)CC(Oc2ccc(O)nn2)c2cc(Br)ccc2O1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
HTT P42858 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7325003 0.84 ABCC9 (0.40) LMNA
SCHEMBL7330893 0.83 TLR3 (0.40) ALDH1A1LMNAHTT
SCHEMBL7326497 0.79 LMNA (0.33) TRPV1ALDH1A1LMNAHTT
SCHEMBL7330531 0.78 ABCC9 (0.38)
SCHEMBL7332017 0.77 ALDH1A1 (0.30) ALDH1A1LMNAHTT
SCHEMBL7331727 0.77 ABCC9 (0.30)
SCHEMBL12315587 0.72 BACE1 (0.32) TRPV1ALDH1A1LMNAHTT
SCHEMBL28768382 0.72 TRPV1 (0.36) TRPV1IDO1
SCHEMBL9141913 0.70 TLR3 (0.43) TRPV1ALDH1A1LMNA
SCHEMBL2184227 0.69 AKR1B1 (0.40) TRPV1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0363883-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1990-04-18 EP disclosed