SCHEMBL7337482

SCHEMBL7337482

COC(=O)Cc1cc(C(F)(F)F)ccc1OCC(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.52
PPARD Q03181 2/20 0.52
PPARA Q07869 2/20 0.52
CYP1A2 P05177 2/20 0.46
CYP2C9 P11712 2/20 0.46
ALDH1A1 P00352 2/20 0.45
CYP2C19 P33261 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HTT P42858 3/20 0.44
KDM4E B2RXH2 3/20 0.44
KMT2A Q03164 2/20 0.44
SSTR4 P31391 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.42
MRGPRX4 Q96LA9 2/20 0.41
FFAR1 O14842 1/20 0.41
FFAR2 O15552 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20576236 0.87 HDAC3 (0.53) PPARGPPARDPPARACYP1A2CYP2C9
SCHEMBL7341566 0.84 PTGDR2 (0.48) PPARGPPARDPPARAHTTKDM4E
SCHEMBL8088577 0.81 L3MBTL1 (0.44) PPARDCYP1A2CYP2C9ALDH1A1HTT
SCHEMBL2858243 0.80 CES2 (0.47) PPARGPPARDPPARAALDH1A1HDAC3
SCHEMBL15524132 0.78 PPARG (0.44) PPARGPPARDPPARACYP1A2CYP2C9
SCHEMBL29331520 0.78 RXRA (0.51) PPARGPPARDPPARACYP1A2CYP2C9
SCHEMBL7040523 0.78 ALDH1A1 (0.44) PPARGPPARDPPARACYP1A2CYP2C9
SCHEMBL18075562 0.77 IDO1 (0.50) PPARGPPARDPPARAALDH1A1KDM4E
SCHEMBL27757329 0.77 ANO1 (0.49) PPARGPPARDPPARAALDH1A1KDM4E
Hydrochloric Acid SCHEMBL7334841 0.76 CYP1A2 (0.47) PPARGPPARDPPARACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed
US-5968938-A Piperazine oxytocin receptor antagonists MERCK & CO., INC. (US) 1999-10-19 US disclosed