SCHEMBL7337997

SCHEMBL7337997

CCCCCC(=O)NCC=Cc1ccc(OCCN2CCOCC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 3/20 0.54
THRA P10827 1/20 0.54
ALDH1A1 P00352 6/20 0.53
LMNA P02545 3/20 0.53
MAPT P10636 1/20 0.53
KMT2A Q03164 1/20 0.53
MAPK1 P28482 2/20 0.52
CYP1A2 P05177 1/20 0.52
CHRM2 P08172 1/20 0.52
CHRM1 P11229 1/20 0.52
HTR2A P28223 1/20 0.52
SCN1A P35498 1/20 0.52
HTR2B P41595 1/20 0.52
KCNH2 Q12809 1/20 0.52
SCN2A Q99250 1/20 0.52
SIGMAR1 Q99720 1/20 0.52
SCN3A Q9NY46 1/20 0.52
HRH3 Q9Y5N1 1/20 0.52
HRH2 P25021 1/20 0.52
HRH1 P35367 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7335005 1.00 THRB (0.54) THRBTHRAALDH1A1LMNAMAPT
SCHEMBL9505612 0.84 THRB (0.63) THRBTHRAALDH1A1LMNAMAPT
SCHEMBL7331718 0.83 HTR1A (0.64) THRBTHRAALDH1A1LMNAMAPT
SCHEMBL14006227 0.79 EPHX2 (0.65) THRBALDH1A1LMNAMAPTKMT2A
SCHEMBL15648875 0.78 ALDH1A1 (0.59) ALDH1A1LMNAMAPK1CYP1A2CHRM2
SCHEMBL15648881 0.78 ALDH1A1 (0.59) ALDH1A1LMNAMAPK1CYP1A2CHRM2
SCHEMBL7335004 0.76 ALDH1A1 (0.51) THRBTHRAALDH1A1LMNAMAPT
SCHEMBL7338002 0.76 THRB (0.53) THRBTHRAALDH1A1LMNAMAPT
SCHEMBL7338536 0.76 ALDH1A1 (0.51) THRBTHRAALDH1A1LMNAMAPT
SCHEMBL7338549 0.76 ALDH1A1 (0.51) THRBTHRAALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0434365-A2 HIV protease inhibitors useful for the treatment of aids MERCK & CO. INC. (US) 1991-06-26 EP claimed
EP-0434365-A2 HIV protease inhibitors useful for the treatment of aids MERCK & CO. INC. (US) 1991-06-26 EP disclosed