SCHEMBL7338201

SCHEMBL7338201

C[n+]1ccn2cc(-c3ccco3)[nH]c(=O)c21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 1/20 0.36
CTSL P07711 1/20 0.36
KDM4E B2RXH2 7/20 0.35
MEN1 O00255 5/20 0.35
KMT2A Q03164 5/20 0.35
MAPT P10636 4/20 0.35
GLA P06280 4/20 0.35
GAA P10253 4/20 0.35
POLB P06746 3/20 0.35
RECQL P46063 3/20 0.35
BLM P54132 3/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
APEX1 P27695 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
ALDH1A1 P00352 3/20 0.34
PKM P14618 1/20 0.34
PLA2G1B P04054 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7327605 0.75 TNKS (0.53) CTSVCTSLKDM4EMEN1KMT2A
SCHEMBL7328378 0.74 TNKS (0.38) KDM4EMEN1KMT2AMAPTL3MBTL1
SCHEMBL7336871 0.72 MAP2K1 (0.44) KDM4EMEN1KMT2AMAPTGLA
SCHEMBL7338197 0.72 CTSV (0.35) CTSVCTSLKDM4EMEN1KMT2A
SCHEMBL7335145 0.71 TNKS (0.56) CTSVCTSLKDM4EMEN1KMT2A
SCHEMBL7337601 0.71 TNKS (0.43) ADORA3
SCHEMBL14469279 0.68 EGFR (0.41) PDE3BPDE3AALDH1A1HPGDADORA1
SCHEMBL27575117 0.62 NOTUM (0.48) CTSVCTSLKDM4EMEN1KMT2A
SCHEMBL11834751 0.62 CTSV (0.44) CTSVCTSLKDM4EMEN1KMT2A
SCHEMBL11835107 0.59 KDM4E (0.58) CTSVCTSLKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726900-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS Aventis Pharma S.A. (FR) 1996-08-21 EP disclosed
WO-1995012594-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1995-05-11 WO disclosed