SCHEMBL7339534

SCHEMBL7339534

CC(C)(C)OC(=O)NCCCCN[C@H](Cc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.54
PRSS1 P07477 1/20 0.54
ACE P12821 2/20 0.54
CMA1 P23946 10/20 0.51
KLK5 Q9Y337 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6412055 0.87 ACE (0.66) F2PRSS1ACECMA1KLK5
SCHEMBL6412059 0.87 ACE (0.66) F2PRSS1ACECMA1KLK5
SCHEMBL7087290 0.87 ACE (0.66) F2PRSS1ACECMA1KLK5
SCHEMBL7343554 0.86 ACE (0.51) F2PRSS1ACE
SCHEMBL7339527 0.83 FKBP1A (0.51) F2PRSS1ACECMA1KLK5
SCHEMBL7339539 0.83 FKBP1A (0.51) F2PRSS1ACECMA1KLK5
SCHEMBL7319098 0.83 ACE (0.51) F2PRSS1ACECMA1KLK5
SCHEMBL7337615 0.82 ITGB3 (0.58) F2PRSS1ACECMA1
SCHEMBL15384069 0.82 KLK5 (0.52) F2PRSS1ACEKLK5
SCHEMBL7337624 0.82 CMA1 (0.45) F2PRSS1ACECMA1KLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5583146-A Heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
EP-0601459-A2 Sulfonamido heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1994-06-15 EP disclosed