SCHEMBL7339539

SCHEMBL7339539

CC(C)(C)OC(=O)NCCCCNC(=O)[C@H]1CCCN1C(=O)[C@H](N)Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 3/20 0.51
CMA1 P23946 7/20 0.51
F2 P00734 2/20 0.51
PRSS1 P07477 1/20 0.51
ACE P12821 1/20 0.50
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49
OPRK1 P41145 1/20 0.49
DPP4 P27487 3/20 0.49
DPP8 Q6V1X1 3/20 0.49
DPP9 Q86TI2 3/20 0.49
DPP7 Q9UHL4 3/20 0.49
FAP Q12884 1/20 0.49
KLK5 Q9Y337 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339527 1.00 FKBP1A (0.51) FKBP1ACMA1F2PRSS1ACE
SCHEMBL7338991 0.85 DPP8 (0.55) FKBP1ACMA1F2PRSS1ACE
SCHEMBL7337615 0.85 ITGB3 (0.58) CMA1F2PRSS1ACE
SCHEMBL7343558 0.84 DPP4 (0.53) FKBP1AF2OPRM1OPRD1OPRK1
SCHEMBL7343548 0.84 DPP4 (0.53) FKBP1AF2OPRM1OPRD1OPRK1
SCHEMBL7339534 0.83 F2 (0.54) CMA1F2PRSS1ACEKLK5
SCHEMBL8366819 0.82 DPP4 (0.58) F2PRSS1ACEOPRM1OPRD1
SCHEMBL7321073 0.82 DPP4 (0.58) F2PRSS1ACEOPRM1OPRD1
SCHEMBL7342500 0.82 PRCP (0.68) FKBP1A
Hydrochloric Acid SCHEMBL11268708 0.82 DPP4 (0.46) FKBP1ACMA1F2PRSS1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5583146-A Heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
EP-0601459-A2 Sulfonamido heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1994-06-15 EP disclosed