SCHEMBL7339727

SCHEMBL7339727

CC(C)CC(N)C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)NC1CN2CCC1CC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IL1RN P18510 1/20 0.48
ERAP2 Q6P179 1/20 0.48
ERAP1 Q9NZ08 1/20 0.48
BDKRB2 P30411 3/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
YAP1 P46937 3/20 0.46
CASP1 P29466 1/20 0.46
CASP3 P42574 1/20 0.46
CASP7 P55210 1/20 0.46
CASP6 P55212 1/20 0.46
CASP8 Q14790 1/20 0.46
MME P08473 1/20 0.45
ACE P12821 1/20 0.45
CPA1 P15085 1/20 0.45
ACE2 Q9BYF1 1/20 0.45
KMT2A Q03164 1/20 0.45
CACNA1B Q00975 2/20 0.44
CTSK P43235 1/20 0.43
OPRK1 P41145 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337924 0.85 YAP1 (0.56) IL1RNERAP2ERAP1MMP9MMP8
SCHEMBL7342359 0.84 YAP1 (0.55) IL1RNERAP2ERAP1MMP9MMP8
SCHEMBL7338585 0.83 UTS2R (0.57)
SCHEMBL7345278 0.83 UTS2R (0.57)
SCHEMBL7339723 0.83 MMP9 (0.44) BDKRB2MMP9MMP8YAP1MME
SCHEMBL7338808 0.83 YAP1 (0.45) IL1RNERAP2ERAP1MMP9MMP8
SCHEMBL7342587 0.82 YAP1 (0.51) IL1RNERAP2ERAP1MMP9MMP8
SCHEMBL7348165 0.81 YAP1 (0.47) IL1RNERAP2ERAP1MMP9MMP8
SCHEMBL7337028 0.81 PSMB1 (0.58) IL1RNERAP2ERAP1MMP9MMP8
SCHEMBL7337109 0.80 YAP1 (0.49) IL1RNERAP2ERAP1YAP1MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US claimed
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed