SCHEMBL7340198

SCHEMBL7340198

NN=CNc1cccc(C(=O)NCC(=O)NC(Cc2ccco2)C(=O)O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
FOLH1 Q04609 2/20 0.43
POLB P06746 3/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 6/20 0.41
HPGD P15428 2/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
RECQL P46063 1/20 0.41
GLA P06280 1/20 0.40
CTSL P07711 1/20 0.39
ITGB3 P05106 3/20 0.39
ITGB1 P05556 3/20 0.39
ITGAV P06756 3/20 0.39
ITGA5 P08648 3/20 0.39
MDM2 Q00987 2/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337769 0.88 POLB (0.44) NPC1RAB9APOLBMAPTPKM
SCHEMBL6775970 0.85 GPR132 (0.49) ITGB3ITGB1ITGAVITGA5MDM2
SCHEMBL6777803 0.84 ITGB1 (0.39) ITGB3ITGB1ITGAVITGA5MDM2
SCHEMBL7342043 0.84 PIN1 (0.55) NPC1RAB9AMAPTITGB3ITGB1
SCHEMBL7836879 0.83 ITGB3 (0.44) ITGB3ITGB1ITGAVITGA5MDM2
SCHEMBL6782093 0.83 ITGB1 (0.41) ITGB3ITGB1ITGAVITGA5MDM2
SCHEMBL3051751 0.83 GPR139 (0.44) CTSLITGB3ITGB1ITGAVITGA5
SCHEMBL7823171 0.83 ITGB3 (0.50) ITGB3ITGB1ITGAVITGA5MDM2
SCHEMBL7347755 0.82 ITGB3 (0.43) FOLH1ITGB3ITGB1ITGAVITGA5
SCHEMBL7838300 0.82 ITGB3 (0.51) CTSLITGB3ITGB1ITGAVITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-B1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2001-07-18 EP claimed
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed