SCHEMBL7340724

SCHEMBL7340724

CC(C[CH]C(=O)NC(Cc1ccc(C=Cc2ccccc2)cc1)C(=O)NC(C)(C)C)C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.43
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
EED O75530 1/20 0.41
CAPN1 P07384 3/20 0.41
CTSB P07858 3/20 0.41
BACE1 P56817 1/20 0.41
EGFR P00533 1/20 0.40
NOS2 P35228 3/20 0.40
NOS3 P29474 2/20 0.40
NOS1 P29475 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343130 0.90 CTSL (0.42) CACNA1BCTSLMMP1FCER2
SCHEMBL7348064 0.90 CTSL (0.42) CACNA1BCTSLMMP1FCER2
SCHEMBL7337043 0.87 ACACB (0.43) CACNA1BCTSL
SCHEMBL7344643 0.85 FFAR1 (0.40) PPARGCACNA1BCTSLMMP1
SCHEMBL7341159 0.85 PTPN1 (0.44) CAPN1CTSBCACNA1BCTSLCTSS
SCHEMBL7338154 0.85 PPARG (0.51) PPARG
SCHEMBL7339993 0.84 CACNA1B (0.35) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7347656 0.84 CACNA1B (0.36) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7348620 0.84 NOS2 (0.37) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7338183 0.81 KMT2A (0.41) CAPN1CTSBCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US claimed
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed