SCHEMBL7340852

SCHEMBL7340852

COC(=O)Cn1c(=O)[nH][nH]c1=O

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
ALDH1A1 P00352 3/20 0.41
HSD17B10 Q99714 2/20 0.41
TSHR P16473 2/20 0.40
KAT2B Q92831 1/20 0.40
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
RCE1 Q9Y256 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14123262 0.83 KDM4E (0.49) KDM4ESMN1; SMN2ALDH1A1HSD17B10TSHR
SCHEMBL24703554 0.79 KDM4E (0.57) KDM4ESMN1; SMN2ALDH1A1HSD17B10TSHR
SCHEMBL7344009 0.79 TSHR (0.46) KDM4ESMN1; SMN2ALDH1A1HSD17B10TSHR
SCHEMBL667246 0.72 KDM4E (0.54) KDM4ESMN1; SMN2ALDH1A1HSD17B10TSHR
SCHEMBL7643580 0.71 SLC9A1 (0.58) KDM4ESMN1; SMN2ALDH1A1HSD17B10TSHR
SCHEMBL5712332 0.70 KDM4E (0.51) KDM4ESMN1; SMN2ALDH1A1HSD17B10TSHR
SCHEMBL23635683 0.70 SMN1; SMN2 (0.44) KDM4ESMN1; SMN2ALDH1A1HSD17B10TP53
SCHEMBL11811656 0.68 KDM4E (0.80) KDM4ESMN1; SMN2ALDH1A1HSD17B10TSHR
SCHEMBL24438895 0.67 ALDH1A1 (0.54) KDM4ESMN1; SMN2ALDH1A1HSD17B10KAT2B
SCHEMBL1006937 0.67 CYP3A4 (0.57) KDM4ESMN1; SMN2ALDH1A1HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4307094-A ANTIHYPERTENSIVE AGENTS HOFFMANN-LA ROCHE INC. (US) 1981-12-22 US disclosed
EP-0024309-A2 Triazolopyridazine derivatives, process and intermediates for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-03-04 EP disclosed