SCHEMBL7340863

SCHEMBL7340863

O=C(Nc1ccc(C(=O)N2Cc3cccnc3Oc3ccccc32)cn1)c1ccccc1-c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.46
CHRNB4 P30926 1/20 0.46
CHRNA3 P32297 1/20 0.46
CHRNA4 P43681 1/20 0.46
AVPR2 P30518 2/20 0.44
OXTR P30559 2/20 0.44
AVPR1A P37288 2/20 0.44
MTTP P55157 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7334184 0.93 TP53 (0.47) CHRNB2CHRNB4CHRNA3CHRNA4AVPR2
SCHEMBL7334422 0.89 TP53 (0.41)
SCHEMBL7342685 0.88 TP53 (0.40)
SCHEMBL7343236 0.88 AVPR2 (0.45) AVPR2AVPR1A
SCHEMBL7345166 0.88 TP53 (0.44)
SCHEMBL7345315 0.87 TP53 (0.40)
SCHEMBL7345024 0.87 AVPR2 (0.45) AVPR2OXTRAVPR1A
SCHEMBL7335374 0.86 CHRNB2 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4AVPR2
SCHEMBL7335173 0.86 LMNA (0.40)
SCHEMBL7334302 0.86 LMNA (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO claimed
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed