SCHEMBL7335173

SCHEMBL7335173

CN(C)c1ccccc1C(=O)Nc1ccc(C(=O)N2Cc3cccnc3Oc3ccccc32)cn1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7334302 0.92 LMNA (0.40) LMNATP53MAPT
SCHEMBL7343236 0.89 AVPR2 (0.45)
SCHEMBL7345315 0.88 TP53 (0.40) TP53MAPT
SCHEMBL7334422 0.88 TP53 (0.41) TP53MAPT
SCHEMBL7342685 0.88 TP53 (0.40) TP53MAPT
SCHEMBL7345166 0.87 TP53 (0.44) TP53MAPT
SCHEMBL7342280 0.87 MEN1 (0.47) TP53
SCHEMBL7340863 0.86 CHRNB2 (0.46)
SCHEMBL7343290 0.85
SCHEMBL7340399 0.85 WNT1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed