SCHEMBL7340982

SCHEMBL7340982

CC(C)[C@H](NC(=O)OCc1cccnc1)C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H](NC(=O)OCc1cccnc1)C(C)C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 4/20 0.57
CYP3A4 P08684 3/20 0.51
CA2 P00918 1/20 0.47
PSMB11 A5LHX3 5/20 0.46
PSMA7 O14818 5/20 0.46
PSMB1 P20618 5/20 0.46
PSMA1 P25786 5/20 0.46
PSMA2 P25787 5/20 0.46
PSMA3 P25788 5/20 0.46
PSMA4 P25789 5/20 0.46
PSMB8 P28062 5/20 0.46
PSMB9 P28065 5/20 0.46
PSMA5 P28066 5/20 0.46
PSMB4 P28070 5/20 0.46
PSMB6 P28072 5/20 0.46
PSMB5 P28074 5/20 0.46
PSMB10 P40306 5/20 0.46
PSMB3 P49720 5/20 0.46
PSMB2 P49721 5/20 0.46
PSMA6 P60900 5/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268971 0.94 CTSD (0.63) CTSDCYP3A4CA2CTSLCTSB
SCHEMBL7275770 0.93 CTSD (0.65) CTSDCYP3A4CA2CTSLCTSB
SCHEMBL6449478 0.93 CTSD (0.63) CTSDCYP3A4CA2CTSLCTSB
SCHEMBL6448343 0.93 CTSD (0.63) CTSDCYP3A4CA2CTSLCTSB
SCHEMBL6446319 0.93 CTSD (0.63) CTSDCYP3A4CA2CTSLCTSB
SCHEMBL6447685 0.87 CTSD (0.57) CTSDCYP3A4CA2CTSLCTSB
SCHEMBL6446462 0.86 CTSD (0.56) CTSDCYP3A4
SCHEMBL7268683 0.86 CTSD (0.65) CTSDCYP3A4CA2PSMB11PSMA7
SCHEMBL7279498 0.85 CTSD (0.60) CTSDCYP3A4CA2GPR132
SCHEMBL7336336 0.85 CA2 (0.60) CTSDCYP3A4CA2CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed