SCHEMBL7341997

SCHEMBL7341997

N#Cc1ccc(N(C(=O)CCl)c2ccccc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.71
RAB9A P51151 8/20 0.71
ALDH1A1 P00352 7/20 0.71
KMT2A Q03164 6/20 0.71
HTT P42858 4/20 0.71
NPSR1 Q6W5P4 4/20 0.71
POLB P06746 1/20 0.71
MEN1 O00255 4/20 0.48
MITF O75030 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
PAX8 Q06710 5/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
LMNA P02545 3/20 0.45
GLA P06280 1/20 0.45
TP53 P04637 1/20 0.45
MAPT P10636 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HKDC1 Q2TB90 1/20 0.43
TSHR P16473 1/20 0.41
SNCA P37840 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2345303 0.84 ALDH1A1 (1.00) NPC1RAB9AALDH1A1KMT2AHTT
SCHEMBL14698064 0.81 KMT2A (0.54) NPC1RAB9AALDH1A1KMT2AHTT
SCHEMBL21800131 0.81 KMT2A (0.51) NPC1RAB9AALDH1A1KMT2AHTT
SCHEMBL7339289 0.78 RAB9A (0.79) NPC1RAB9AALDH1A1KMT2AHTT
SCHEMBL31393776 0.77 KMT2A (0.57) NPC1RAB9AALDH1A1KMT2ANPSR1
SCHEMBL31074337 0.77 FNIP1 (0.60) NPC1RAB9AALDH1A1KMT2AHTT
SCHEMBL27534539 0.75 KMT2A (0.49) NPC1ALDH1A1KMT2AHTTMEN1
SCHEMBL2112731 0.75 KMT2A (0.63) NPC1ALDH1A1KMT2ANPSR1MEN1
SCHEMBL7338508 0.74 NPC1 (0.71) NPC1RAB9AALDH1A1KMT2AHTT
SCHEMBL7339671 0.74 CACNA2D1 (0.53) NPC1RAB9AALDH1A1HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0658157-A1 DIARYL PIPERAZINOACETAMIDE COMPOUNDS AS ANTIMUSCARINIC AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-06-21 EP disclosed
WO-1994005648-A1 DIARYL PIPERAZINOACETAMIDE COMPOUNDS AS ANTIMUSCARINIC AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-17 WO disclosed
EP-0585500-A1 Diaryl piperazineacetamides as antimuscarinic agents MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-09 EP disclosed