SCHEMBL7342953

SCHEMBL7342953

CC(C)(C)ON1CCC(Oc2ccc(CBr)c(OC(F)(F)F)c2)CC1=C=O

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OXTR P30559 1/20 0.36
EPHX2 P34913 2/20 0.33
UTS2R Q9UKP6 3/20 0.32
SCN9A Q15858 3/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2J2 P51589 1/20 0.31
MCHR1 Q99705 1/20 0.31
MGLL Q99685 1/20 0.30
LIPE Q05469 2/20 0.30
GPR119 Q8TDV5 1/20 0.30
HTR2A P28223 2/20 0.30
ACACB O00763 1/20 0.30
MMP12 P39900 1/20 0.30
MMP13 P45452 1/20 0.30
MMP14 P50281 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7335906 0.91 OXTR (0.37) OXTREPHX2SCN9ACYP2C9CYP2J2
SCHEMBL7342824 0.88 OXTR (0.40) OXTREPHX2SCN9ACYP2C9CYP2J2
SCHEMBL8092927 0.87 EPHX2 (0.37) EPHX2UTS2R
SCHEMBL8088578 0.80 EPHX2 (0.40) EPHX2GPR119
SCHEMBL7343847 0.79
SCHEMBL7333661 0.78 OXTR (0.42) OXTRLIPEGPR119ACACB
SCHEMBL8088615 0.78 EPHX2 (0.36) EPHX2GPR119
SCHEMBL8081388 0.77 EPHX2 (0.40) EPHX2LIPEGPR119
SCHEMBL7335803 0.77 GPR119 (0.52) OXTREPHX2LIPEGPR119
SCHEMBL7333820 0.77 OXTR (0.41) OXTREPHX2SCN9ACYP2C9MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed
US-5968938-A Piperazine oxytocin receptor antagonists MERCK & CO., INC. (US) 1999-10-19 US disclosed