SCHEMBL7343547

SCHEMBL7343547

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2Cc3ccccc3C2)C1c1ccccc1Br

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.47
CYP2C9 P11712 4/20 0.47
CYP1A2 P05177 4/20 0.47
HSD17B10 Q99714 4/20 0.47
KDM4E B2RXH2 3/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C19 P33261 3/20 0.47
KMT2A Q03164 3/20 0.47
HIF1A Q16665 3/20 0.47
ABCB11 O95342 3/20 0.47
LMNA P02545 3/20 0.47
SCN1A P35498 3/20 0.47
SCN5A Q14524 3/20 0.47
SCN2A Q99250 3/20 0.47
SCN3A Q9NY46 3/20 0.47
NR1I2 O75469 3/20 0.47
MEN1 O00255 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
TP53 P04637 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349519 0.88 ADORA3 (0.57) ADORA3CYP2C9CYP1A2HSD17B10KDM4E
SCHEMBL7348023 0.88 CACNA1C (0.48) ADORA3CYP2C9CYP1A2HSD17B10KDM4E
SCHEMBL7351367 0.85 ADORA3 (0.69) ADORA3CYP2C9CYP1A2HSD17B10KDM4E
SCHEMBL7347553 0.83 KDM4E (0.59) ADORA3CYP2C9CYP1A2HSD17B10KDM4E
SCHEMBL7345495 0.83 POLB (0.58) ADORA3CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7350408 0.83 PDE1C (0.69) ADORA3CYP2C9CYP1A2HSD17B10KDM4E
SCHEMBL7340139 0.82 ADORA3 (0.47) ADORA3CYP2C9CYP1A2HSD17B10KDM4E
SCHEMBL7344861 0.82 HSD17B10 (0.66) ADORA3CYP2C9CYP1A2HSD17B10KDM4E
SCHEMBL7342397 0.82 ADORA3 (0.47) ADORA3CYP2C9CYP1A2HSD17B10KDM4E
SCHEMBL3034394 0.81 ADORA3 (0.68) ADORA3CYP2C9CYP1A2HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed