SCHEMBL7347553

SCHEMBL7347553

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2Cc3ccccc3C2)C1c1ccc(Br)o1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.59
NPSR1 Q6W5P4 2/20 0.59
POLB P06746 1/20 0.59
GPR55 Q9Y2T6 1/20 0.59
ADORA3 P0DMS8 1/20 0.44
MAPT P10636 6/20 0.43
ALDH1A1 P00352 4/20 0.43
HPGD P15428 2/20 0.43
HTT P42858 1/20 0.43
CACNA1F O60840 1/20 0.41
CACNA1D Q01668 1/20 0.41
CACNA1S Q13698 1/20 0.41
CACNA1C Q13936 1/20 0.41
HSD17B10 Q99714 2/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7347855 0.85 MAPT (0.51) KDM4ENPSR1POLBADORA3MAPT
SCHEMBL7349712 0.85 KDM4E (0.67) KDM4ENPSR1POLBADORA3MAPT
SCHEMBL7343547 0.83 ADORA3 (0.47) KDM4ENPSR1ADORA3MAPTALDH1A1
SCHEMBL7341163 0.83 HSD17B10 (0.63) KDM4ENPSR1POLBGPR55ADORA3
SCHEMBL7347558 0.82 KDM4E (0.72) KDM4ENPSR1POLBGPR55ADORA3
SCHEMBL7345495 0.81 POLB (0.58) NPSR1POLBGPR55ADORA3MAPT
SCHEMBL7347551 0.81 KDM4E (0.53) KDM4ENPSR1POLBGPR55ADORA3
SCHEMBL7347564 0.80 KDM4E (0.55) KDM4ENPSR1POLBGPR55ADORA3
SCHEMBL7340139 0.80 ADORA3 (0.47) KDM4EADORA3MAPTALDH1A1HPGD
SCHEMBL7342397 0.80 ADORA3 (0.47) KDM4EADORA3MAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed